SCHEMBL24329591

SCHEMBL24329591

COC(=O)c1ccc2nc(CN3CCC(c4cccc(OCc5cc(C)c(C(=O)C6CC6)cc5F)n4)CC3)n(CC3CCO3)c2c1

nearest known ligand 0.75

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GLP1R P43220 20/20 0.75
CYP2C8 P10632 2/20 0.66
KCNH2 Q12809 2/20 0.66
HTR1A P08908 1/20 0.66
HTR2A P28223 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29053111 1.00 GLP1R (0.75) GLP1RCYP2C8KCNH2HTR1AHTR2A
SCHEMBL29053074 0.95 GLP1R (0.73) GLP1RCYP2C8KCNH2HTR1AHTR2A
SCHEMBL25957684 0.95 GLP1R (0.73) GLP1RCYP2C8KCNH2HTR1AHTR2A
SCHEMBL29555218 0.94 GLP1R (0.85) GLP1RCYP2C8KCNH2HTR1AHTR2A
SCHEMBL24330495 0.94 GLP1R (0.85) GLP1RCYP2C8KCNH2HTR1AHTR2A
SCHEMBL24329478 0.94 GLP1R (0.85) GLP1RCYP2C8KCNH2HTR1AHTR2A
SCHEMBL29555016 0.94 GLP1R (0.85) GLP1RCYP2C8KCNH2HTR1AHTR2A
SCHEMBL24329497 0.93 GLP1R (0.87) GLP1RCYP2C8KCNH2HTR1AHTR2A
SCHEMBL29555267 0.93 GLP1R (0.87) GLP1RCYP2C8KCNH2HTR1AHTR2A
SCHEMBL29053081 0.93 GLP1R (0.87) GLP1RCYP2C8KCNH2HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4227299-A1 BENZIMIDAZOLONE GLP-1 RECEPTOR AGONIST AND USE THEREOF Hangzhou Zhongmeihuadong Pharmaceutical Co., Ltd. (CN) 2023-08-16 EP disclosed
CN-116348464-A Benzimidazolone GLP-1 receptor agonists and uses thereof 杭州中美华东制药有限公司 2023-06-27 CN disclosed
WO-2022078152-A1 BENZIMIDAZOLONE GLP-1 RECEPTOR AGONIST AND USE THEREOF 杭州中美华东制药有限公司 2022-04-21 WO disclosed