SCHEMBL24363496

SCHEMBL24363496

Nc1ncnc(NC2CCCCC2)c1-c1ccc(Oc2ccccc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 16/20 0.68
KCNH2 Q12809 3/20 0.66
EGFR P00533 3/20 0.65
TEC P42680 1/20 0.52
BMX P51813 1/20 0.52
CD69 Q07108 1/20 0.52
ITK Q08881 1/20 0.52
ERBB4 Q15303 1/20 0.52
GP6 Q9HCN6 1/20 0.52
NUDT5 Q9UKK9 1/20 0.52
LCK P06239 6/20 0.51
KDR P35968 5/20 0.51
TEK Q02763 5/20 0.51
LYN P07948 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
RGS12 O14924 1/20 0.50
NPC1 O15118 1/20 0.50
GMNN O75496 1/20 0.50
ALDH1A1 P00352 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24363230 0.99 BTK (0.69) BTKKCNH2EGFRTECBMX
SCHEMBL14165691 0.89 BTK (0.70) BTKKCNH2EGFRTECBMX
SCHEMBL20480850 0.89 BTK (0.70) BTKKCNH2EGFRTECBMX
SCHEMBL14165704 0.89 BTK (0.70) BTKKCNH2EGFRTECBMX
SCHEMBL14165430 0.88 BTK (0.66) BTKKCNH2EGFRTECBMX
SCHEMBL14165553 0.87 BTK (0.60) BTKKCNH2EGFRTECBMX
SCHEMBL14165937 0.87 BTK (0.60) BTKKCNH2EGFRTECBMX
SCHEMBL24363262 0.87 BTK (0.68) BTKKCNH2EGFRTECBMX
SCHEMBL14165552 0.87 BTK (0.60) BTKKCNH2EGFRTECBMX
SCHEMBL23722580 0.85 BTK (0.74) BTKKCNH2EGFRTECBMX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2718270-B1 COMPOSITIONS AND METHODS FOR THE PRODUCTION OF PYRIMIDINE AND PYRIDINE COMPOUNDS WITH BTK INHIBITORY ACTIVITY MERCK PATENT GMBH (DE) 2022-04-27 EP disclosed