SCHEMBL24364796

SCHEMBL24364796

COCc1ccc([C@H]2CC[C@H](C)CN2)cc1

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.32
REN P00797 2/20 0.32
ESR2 Q92731 1/20 0.32
BRD4 O60885 1/20 0.32
CREBBP Q92793 1/20 0.32
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24364795 0.81 ESR2 (0.33) ESR2
SCHEMBL25322649 0.79 HRH3 (0.41)
SCHEMBL25322631 0.79 KCNH2 (0.54) KCNH2PTGS2
SCHEMBL25322627 0.79 KCNH2 (0.54) KCNH2PTGS2
SCHEMBL31145247 0.78 ESR2 (0.53) ESR2
SCHEMBL29324808 0.78 ESR2 (0.53) ESR2
SCHEMBL24364303 0.78 ESR2 (0.53) ESR2
SCHEMBL25321512 0.76 MAPT (0.39) ESR2
SCHEMBL24233794 0.76 MAPT (0.39) ESR2
SCHEMBL14963942 0.76 MAPT (0.39) ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220127256-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. 2022-04-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220127256-A1 COMPOUNDS AND METHODS OF USE F12, C1R, ABCG2 KCNH2 1114/4885REN 19/4885ESR2 935/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.