SCHEMBL24376705

SCHEMBL24376705

Cc1cc2c(cc1Sc1nc3c(N)ncnc3n1CCCS(=O)(=O)NCC(C)C)C(=O)CC2

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 11/20 0.48
HSP90AB1 P08238 10/20 0.48
HSP90B1 P14625 12/20 0.47
TRAP1 Q12931 7/20 0.47
ERBB2 P04626 7/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15609910 0.92 HSP90AB1 (0.51) HSP90AA1HSP90AB1HSP90B1TRAP1ERBB2
SCHEMBL29580667 0.92 HSP90AB1 (0.51) HSP90AA1HSP90AB1HSP90B1TRAP1ERBB2
SCHEMBL24377228 0.89 HSP90AA1 (0.48) HSP90AA1HSP90AB1HSP90B1TRAP1ERBB2
SCHEMBL24376805 0.89 HSP90AB1 (0.51) HSP90AA1HSP90AB1HSP90B1TRAP1ERBB2
SCHEMBL24376810 0.89 HSP90B1 (0.49) HSP90AA1HSP90AB1HSP90B1TRAP1ERBB2
SCHEMBL24376800 0.88 HSP90AA1 (0.51) HSP90AA1HSP90AB1HSP90B1TRAP1ERBB2
SCHEMBL24376781 0.88 HSP90AA1 (0.49) HSP90AA1HSP90AB1HSP90B1TRAP1ERBB2
SCHEMBL24376701 0.88 HSP90AA1 (0.50) HSP90AA1HSP90AB1HSP90B1TRAP1ERBB2
SCHEMBL24376782 0.87 HSP90AA1 (0.48) HSP90AA1HSP90AB1HSP90B1TRAP1ERBB2
SCHEMBL13193749 0.87 ERBB2 (0.49) HSP90AA1HSP90AB1HSP90B1TRAP1ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2694505-B1 HSP90 INHIBITORS SLOAN KETTERING INST CANCER RES (US) 2022-04-27 EP disclosed