SCHEMBL24376834

SCHEMBL24376834

CCc1cc2c(cc1Sc1nc3c(N)ncnc3n1CCS(=O)(=O)NC1CC1)C(F)CC2

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 18/20 0.40
HSP90AB1 P08238 18/20 0.40
ERBB2 P04626 3/20 0.38
HSP90B1 P14625 2/20 0.38
TRAP1 Q12931 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24377269 0.92 HSP90AA1 (0.41) HSP90AA1HSP90AB1ERBB2HSP90B1TRAP1
SCHEMBL24377264 0.90 HSP90AA1 (0.42) HSP90AA1HSP90AB1ERBB2HSP90B1TRAP1
SCHEMBL15609921 0.90 HSP90AB1 (0.44) HSP90AA1HSP90AB1ERBB2HSP90B1TRAP1
SCHEMBL24377286 0.89 HSP90AA1 (0.51) HSP90AA1HSP90AB1ERBB2HSP90B1TRAP1
SCHEMBL24376769 0.88 HSP90AA1 (0.42) HSP90AA1HSP90AB1ERBB2HSP90B1TRAP1
SCHEMBL24376906 0.87 HSP90B1 (0.47) HSP90AA1HSP90AB1ERBB2HSP90B1TRAP1
SCHEMBL24376870 0.87 HSP90AA1 (0.41) HSP90AA1HSP90AB1ERBB2HSP90B1TRAP1
SCHEMBL24377304 0.86 HSP90AA1 (0.43) HSP90AA1HSP90AB1ERBB2HSP90B1
SCHEMBL24376762 0.86 HSP90AA1 (0.45) HSP90AA1HSP90AB1ERBB2HSP90B1TRAP1
SCHEMBL24377278 0.85 HSP90AA1 (0.42) HSP90AA1HSP90AB1ERBB2HSP90B1TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2694505-B1 HSP90 INHIBITORS SLOAN KETTERING INST CANCER RES (US) 2022-04-27 EP disclosed