SCHEMBL24376907

SCHEMBL24376907

CCc1cc2c(cc1Sc1nc3c(N)ncnc3n1CCNC(=O)C(C)(C)C)C(F)CC2

nearest known ligand 0.44

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 20/20 0.44
HSP90AA1 P07900 19/20 0.44
ERBB2 P04626 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15609465 0.91 HSP90AB1 (0.49) HSP90AB1HSP90AA1ERBB2
SCHEMBL24376908 0.90 HSP90AA1 (0.44) HSP90AB1HSP90AA1
SCHEMBL24376836 0.87 HSP90AA1 (0.51) HSP90AB1HSP90AA1ERBB2
SCHEMBL24377281 0.87 HSP90AA1 (0.44) HSP90AB1HSP90AA1
SCHEMBL24376826 0.86 HSP90AA1 (0.45) HSP90AB1HSP90AA1
SCHEMBL24376870 0.85 HSP90AA1 (0.41) HSP90AB1HSP90AA1ERBB2
SCHEMBL24377304 0.85 HSP90AA1 (0.43) HSP90AB1HSP90AA1ERBB2
SCHEMBL24377269 0.85 HSP90AA1 (0.41) HSP90AB1HSP90AA1ERBB2
SCHEMBL24377278 0.84 HSP90AA1 (0.42) HSP90AB1HSP90AA1ERBB2
SCHEMBL24376711 0.84 HSP90AB1 (0.52) HSP90AB1HSP90AA1ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2694505-B1 HSP90 INHIBITORS SLOAN KETTERING INST CANCER RES (US) 2022-04-27 EP disclosed