SCHEMBL24399063

SCHEMBL24399063

C#Cc1cc2ncnc(Nc3cccc(Cl)c3F)c2cc1NC(=O)/C=C/CN1CCOCC1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.56
ERBB2 P04626 11/20 0.56
ERBB4 Q15303 6/20 0.56
JAK3 P52333 1/20 0.56
KCNH2 Q12809 1/20 0.56
ERBB3 P21860 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22983382 0.86 EGFR (0.51) EGFRERBB2ERBB4JAK3KCNH2
SCHEMBL29718961 0.86 EGFR (0.51) EGFRERBB2ERBB4JAK3KCNH2
SCHEMBL22983387 0.86 EGFR (0.51) EGFRERBB2ERBB4JAK3KCNH2
SCHEMBL17200124 0.86 EGFR (0.63) EGFRERBB2ERBB4JAK3KCNH2
SCHEMBL17200125 0.86 EGFR (0.63) EGFRERBB2ERBB4JAK3KCNH2
SCHEMBL31638765 0.85 EGFR (0.48) EGFRERBB2ERBB4JAK3KCNH2
SCHEMBL24398908 0.84 EGFR (0.49) EGFRERBB2ERBB4JAK3KCNH2
SCHEMBL24398880 0.84 EGFR (0.49) EGFRERBB2ERBB4JAK3KCNH2
SCHEMBL22983932 0.84 EGFR (0.49) EGFRERBB2ERBB4JAK3KCNH2
SCHEMBL31638901 0.84 EGFR (0.48) EGFRERBB2ERBB4JAK3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022094464-A1 METHOD OF TREATING CANCERS WITH ALKYNE SUBSTITUTED QUINAZOLINE DERIVATIVES BLACK DIAMOND THERAPEUTICS, INC. (US) 2022-05-05 WO disclosed