SCHEMBL24424865

SCHEMBL24424865

Cc1c(Cl)cnc(C#N)c1F

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
POLB P06746 1/20 0.46
CYP11B2 P19099 1/20 0.33
DAO P14920 1/20 0.33
PLAU P00749 1/20 0.33
GRM5 P41594 1/20 0.31
USP8 P40818 1/20 0.30
USP7 Q93009 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2297778 0.81 KDM4E (0.46) KDM4EALDH1A1POLBCYP11B2GRM5
SCHEMBL20113370 0.80 USP8 (0.35) KDM4EALDH1A1POLBCYP11B2DAO
SCHEMBL18283690 0.80 POLB (0.48) KDM4EALDH1A1POLBDAOPLAU
SCHEMBL29368821 0.80 USP8 (0.35) KDM4EALDH1A1POLBCYP11B2DAO
SCHEMBL18283565 0.80 POLB (0.48) KDM4EALDH1A1POLBDAOPLAU
SCHEMBL31410007 0.73 DAO (0.37) ALDH1A1DAOPLAU
SCHEMBL31409944 0.72
SCHEMBL29877981 0.71 KDM4E (0.32) KDM4EALDH1A1POLB
SCHEMBL22976756 0.70 KDM4E (0.40) KDM4EALDH1A1POLBCYP11B2GRM5
SCHEMBL2220883 0.69 PLAU (0.39) ALDH1A1DAOPLAUUSP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220144802-A1 NONPEPTIDE SOMATOSTATIN TYPE 5 RECEPTOR AGONISTS AND USES THEREOF Crinetics Pharmaceuticals, Inc. 2022-05-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220144802-A1 NONPEPTIDE SOMATOSTATIN TYPE 5 RECEPTOR AGONISTS AND USES THEREOF SSTR5, SSTR4, SSTR3 KDM4E 4514/4885ALDH1A1 4555/4885POLB 4524/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.