SCHEMBL24428847

SCHEMBL24428847

C[C@H]1C[C@@H](Cc2ccc(-c3cc(Cl)ccc3F)cc2)NC1=O

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.39
FFAR4 Q5NUL3 3/20 0.38
ROCK1 Q13464 2/20 0.37
MAOB P27338 1/20 0.35
GRM2 Q14416 3/20 0.35
HTR2A P28223 2/20 0.34
MME P08473 3/20 0.34
ACE P12821 1/20 0.34
GHSR Q92847 1/20 0.34
FASN P49327 1/20 0.33
FFAR1 O14842 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20364012 0.84 MAOB (0.39) ROCK2FFAR4ROCK1MAOBHTR2A
SCHEMBL20364020 0.82 MME (0.36) ROCK2FFAR4ROCK1MAOBMME
SCHEMBL24380861 0.82 MME (0.36) ROCK2FFAR4ROCK1MAOBMME
SCHEMBL16979073 0.80 CHRM1 (0.37) ROCK2FFAR4MAOBHTR2AFASN
SCHEMBL16979069 0.78 KCNA5 (0.43) ROCK2MAOB
SCHEMBL10847469 0.78 GAA (0.48) GHSR
SCHEMBL8283063 0.78 GAA (0.48) GHSR
SCHEMBL1908538 0.75 GRM2 (0.40) ROCK2GRM2
SCHEMBL20072321 0.75 GRM2 (0.40) ROCK2GRM2
SCHEMBL4440151 0.75 GRM2 (0.40) ROCK2GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3256446-B1 (2S,4R)-5-(5'-CHLORO-2'-FLUOROBIPHENYL-4-YL)-4-(ETHOXYOXALYLAMINO)-2-HYDROXYMETHYL-2-METHYLPENTANOIC ACID AS NEPRILYSIN INHIBITOR THERAVANCE BIOPHARMA R&D IP LLC (US) 2022-05-18 EP disclosed