SCHEMBL2443349

SCHEMBL2443349

O=C(Nc1noc2ccccc12)c1cccc(F)c1F.O=C([15NH]c1noc2ccccc12)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 8/20 0.60
TP53 P04637 7/20 0.60
MAPT P10636 3/20 0.49
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
KCNJ6 P48051 1/20 0.42
KCNJ3 P48549 1/20 0.42
ACHE P22303 1/20 0.41
MAOB P27338 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
HIF1A Q16665 2/20 0.40
KCNJ11 Q14654 1/20 0.39
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
PKM P14618 1/20 0.38
RAB9A P51151 1/20 0.38
CSF1R P07333 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2442472 0.87 TP53 (0.66) SMN1; SMN2TP53MAPTALOX15TSHR
SCHEMBL2442817 0.87 SMN1; SMN2 (0.76) SMN1; SMN2TP53MAPTMEN1KMT2A
SCHEMBL2443302 0.78 TP53 (0.74) SMN1; SMN2TP53MAPTALOX15TSHR
SCHEMBL2439106 0.77 SMN1; SMN2 (0.58) SMN1; SMN2TP53MAPTMEN1KMT2A
SCHEMBL2438649 0.76 SMN1; SMN2 (0.54) SMN1; SMN2TP53MAPTKMT2ACSF1R
SCHEMBL2439676 0.76 TP53 (0.54) SMN1; SMN2TP53MAPTMAOBMEN1
SCHEMBL2442316 0.75 TP53 (1.00) SMN1; SMN2TP53MAPTMEN1KMT2A
SCHEMBL2439755 0.73 TP53 (0.66) SMN1; SMN2TP53MAPTALOX15TSHR
SCHEMBL2441769 0.73 MEN1 (0.48) SMN1; SMN2TP53MAPTACHEMAOB
SCHEMBL2438675 0.72 TP53 (0.82) SMN1; SMN2TP53MAPTALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893589-B1 SUBSTITUTED N-BENZO [D] ISOXAZOL-3-YL-AMINE DERIVATIVES AS INHIBITORS OF MGLUR5, SEROTONINE (5-HT) AND NORADRENALINE RECEPTORS, AND THE USE THEREOF FOR PRODUCING MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-09-14 EP claimed