SCHEMBL24438005

SCHEMBL24438005

Cn1cc(-c2cn3nc(NC(=O)OC(C)(C)C)cc3c(O)n2)cn1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.53
DYRK1A Q13627 3/20 0.53
TTK P33981 10/20 0.41
RET P07949 5/20 0.38
S1PR2 O95136 1/20 0.38
CCNA2 P20248 2/20 0.37
CDK2 P24941 2/20 0.37
AURKA O14965 1/20 0.37
WNT1 P04628 1/20 0.37
NTRK1 P04629 1/20 0.37
EPHB2 P29323 1/20 0.37
KDR P35968 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24438647 0.79 DYRK1A (0.43) GSK3BDYRK1ATTKRETCCNA2
SCHEMBL27170240 0.77 BTK (0.54) GSK3BDYRK1ATTKRETCCNA2
SCHEMBL24437819 0.77 BTK (0.54) GSK3BDYRK1ATTKRETCCNA2
SCHEMBL27170238 0.77 BTK (0.54) GSK3BDYRK1ATTKRETCCNA2
SCHEMBL25236672 0.76 CHEK1 (0.39) KDRIRAK4
SCHEMBL17801236 0.74 CHEK1 (0.47) IRAK4
SCHEMBL20967198 0.74 DYRK1A (0.75) GSK3BDYRK1AWNT1
SCHEMBL19253504 0.74 JAK2 (0.48) KDR
SCHEMBL24438255 0.73 JAK2 (0.41) TTKAURKAKDR
SCHEMBL24060899 0.72 ERN1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022104079-A1 PYRAZOLO[1,5-A]PYRAZINE DERIVATIVES AS BTK INHIBITORS BIOGEN MA INC. (US) 2022-05-19 WO disclosed