SCHEMBL24439620

SCHEMBL24439620

COC(=O)[C@H]1CCC[C@H](Oc2ccc(-c3sc(F)cc3C=O)nc2C)C1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 5/20 0.40
ABCC3 O15438 2/20 0.37
ABCC4 O15439 2/20 0.37
SLCO1B3 Q9NPD5 2/20 0.37
SLCO1B1 Q9Y6L6 2/20 0.37
ABCB11 O95342 1/20 0.37
FFAR4 Q5NUL3 3/20 0.33
PI4KB Q9UBF8 2/20 0.33
PDE4B Q07343 3/20 0.33
PDE4A P27815 2/20 0.33
PDE4C Q08493 2/20 0.33
PDE4D Q08499 2/20 0.33
TMPRSS15 P98073 1/20 0.31
HCRTR1 O43613 2/20 0.31
HCRTR2 O43614 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24439392 1.00 LPAR1 (0.40) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL29517764 1.00 LPAR1 (0.40) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL29577128 0.91 LPAR1 (0.41) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL28744990 0.91 LPAR1 (0.46) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL24441674 0.91 LPAR1 (0.41) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL24441049 0.89 LPAR1 (0.40) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL29576333 0.89 LPAR1 (0.40) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL24440690 0.89 LPAR1 (0.40) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL29576361 0.89 LPAR1 (0.40) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL24439618 0.87 LPAR1 (0.41) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022100624-A1 OXY-SUBSTITUTED AMINOCARBONATE THIOPHENE-BASED COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed
WO-2022100623-A1 NITROGEN-SUBSTITUTED HETEROCYCLIC THIOPHENE COMPOUNDS AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed
WO-2022100623-A1 NITROGEN-SUBSTITUTED HETEROCYCLIC THIOPHENE COMPOUNDS AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed
CN-114456159-A Nitrogen-substituted heterocyclic thiophene compound and application thereof 武汉人福创新药物研发中心有限公司 2022-05-10 CN disclosed