SCHEMBL24439677

SCHEMBL24439677

COC(=O)[C@H]1CCC[C@H](Oc2ccc(-c3sc(Cl)cc3COC(=O)NCCC3CC3)nc2C)C1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 6/20 0.38
ABCC3 O15438 2/20 0.38
ABCC4 O15439 2/20 0.38
SLCO1B3 Q9NPD5 2/20 0.38
SLCO1B1 Q9Y6L6 2/20 0.38
ABCB11 O95342 1/20 0.38
SCD O00767 1/20 0.32
PI4KB Q9UBF8 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29672272 0.93 LPAR1 (0.44) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL29518045 0.93 SLCO1B1 (0.40) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL24439788 0.93 SLCO1B1 (0.40) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL24439699 0.90 SCD (0.35) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL24439679 0.89 SCD (0.35) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL24439469 0.87 LPAR1 (0.38) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL29517743 0.87 SLCO1B1 (0.47) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL29672231 0.86 SLCO1B1 (0.47) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL24439384 0.86 SLCO1B1 (0.47) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL24441591 0.85 LPAR1 (0.39) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022100624-A1 OXY-SUBSTITUTED AMINOCARBONATE THIOPHENE-BASED COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed
WO-2022100624-A1 OXY-SUBSTITUTED AMINOCARBONATE THIOPHENE-BASED COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed
CN-114456147-A Oxygen substituted amino carbonate thiophene compounds 武汉人福创新药物研发中心有限公司 2022-05-10 CN disclosed