SCHEMBL24439733

SCHEMBL24439733

COC(=O)[C@H]1CCC[C@H](Oc2ccc(-c3sc(Cl)cc3CO)nc2C)C1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 2/20 0.41
ABCC3 O15438 2/20 0.38
ABCC4 O15439 2/20 0.38
SLCO1B3 Q9NPD5 2/20 0.38
SLCO1B1 Q9Y6L6 2/20 0.38
ABCB11 O95342 1/20 0.38
PI4KB Q9UBF8 2/20 0.32
KMO O15229 2/20 0.32
SAE1 Q9UBE0 1/20 0.32
PIK3CD O00329 1/20 0.31
PIK3CG P48736 1/20 0.31
PDE4A P27815 5/20 0.31
PDE4B Q07343 5/20 0.31
PDE4C Q08493 5/20 0.31
PDE4D Q08499 5/20 0.31
CFTR P13569 2/20 0.31
POLB P06746 1/20 0.30
OPRK1 P41145 1/20 0.30
WDR5 P61964 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29625494 1.00 LPAR1 (0.41) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL29625495 0.93 LPAR1 (0.41) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL24441135 0.93 LPAR1 (0.41) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL29625478 0.92 LPAR1 (0.40) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL24441476 0.92 LPAR1 (0.40) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL28745055 0.92 LPAR1 (0.40) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL29576756 0.92 LPAR1 (0.40) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL24441477 0.91 LPAR1 (0.41) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL29576267 0.91 LPAR1 (0.41) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1
SCHEMBL28744676 0.91 LPAR1 (0.47) LPAR1ABCC3ABCC4SLCO1B3SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022100624-A1 OXY-SUBSTITUTED AMINOCARBONATE THIOPHENE-BASED COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed
WO-2022100623-A1 NITROGEN-SUBSTITUTED HETEROCYCLIC THIOPHENE COMPOUNDS AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-05-19 WO disclosed