SCHEMBL24444

SCHEMBL24444

Cc1cccc(Nc2nccn3nc(N(C)c4ccc(Sc5nccn5C)c(Cl)c4)nc23)c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
IGF1R P08069 5/20 0.37
MAP2K1 Q02750 9/20 0.37
KIT P10721 1/20 0.36
PDGFRA P16234 1/20 0.36
KDR P35968 1/20 0.36
LMNA P02545 2/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
HPGD P15428 1/20 0.34
ATM Q13315 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
EGFR P00533 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15216750 0.84 NPC1 (0.45) NPC1RAB9ASMN1; SMN2IGF1RMAP2K1
SCHEMBL15208567 0.78 IGF1R (0.43) IGF1RMAP2K1KDREGFR
SCHEMBL23678 0.78 IGF1R (0.44) IGF1RMAP2K1
SCHEMBL15216751 0.76 IGF1R (0.44) IGF1RMAP2K1LMNAUSP2ALDH1A1
SCHEMBL15206974 0.74 NPC1 (0.43) NPC1RAB9ASMN1; SMN2IGF1RMAP2K1
SCHEMBL24518 0.74 GCK (0.44) SMN1; SMN2IGF1RMAP2K1ALDH1A1TP53
SCHEMBL24626 0.73 IGF1R (0.37) NPC1RAB9ASMN1; SMN2IGF1RMAP2K1
SCHEMBL15206972 0.72 NPC1 (0.43) NPC1RAB9ASMN1; SMN2IGF1RMAP2K1
SCHEMBL24060 0.70 IGF1R (0.47) NPC1RAB9AIGF1RMAP2K1EGFR
SCHEMBL24767 0.70 IGF1R (0.47) NPC1RAB9AIGF1RMAP2K1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012025186-A1 TRIAZOLOPYRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2012-03-01 WO disclosed