SCHEMBL2445978

SCHEMBL2445978

CC(C)(C)OC(=O)N1CC2CCC[C@@H]2C1CNC(=O)c1cnc2sccn12

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 1/20 0.35
RORC P51449 1/20 0.35
HCRTR1 O43613 11/20 0.34
HCRTR2 O43614 4/20 0.34
NAMPT P43490 4/20 0.33
KDM4E B2RXH2 2/20 0.32
PKM P14618 1/20 0.32
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
RECQL P46063 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL497312 1.00 ACKR3 (0.35) ACKR3RORCHCRTR1HCRTR2NAMPT
SCHEMBL496343 0.87 HCRTR1 (0.35) ACKR3RORCHCRTR1HCRTR2NAMPT
SCHEMBL2447646 0.84 HCRTR1 (0.45) HCRTR1HCRTR2
SCHEMBL496234 0.84 HCRTR1 (0.45) HCRTR1HCRTR2
SCHEMBL1340238 0.74 HCRTR1 (0.54) RORCHCRTR1HCRTR2
SCHEMBL2930753 0.74 HCRTR1 (0.54) RORCHCRTR1HCRTR2
SCHEMBL3415424 0.74 HCRTR1 (0.54) RORCHCRTR1HCRTR2
SCHEMBL2930755 0.74 HCRTR1 (0.54) RORCHCRTR1HCRTR2
SCHEMBL1338342 0.74 KIT (0.40) ACKR3RORCNAMPTKDM4EPKM
SCHEMBL3641229 0.72 ACKR3 (0.40) ACKR3HCRTR1KDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164847-B1 3-AZA-BICYCLO[3.3.0]OCTANE COMPOUNDS ACTELION PHARMACEUTICALS LTD (CH) 2011-09-14 EP disclosed