SCHEMBL2446475

SCHEMBL2446475

NC(=O)C1CCCN(c2ccccc2)C1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.62
MEN1 O00255 1/20 0.62
NOTUM Q6P988 1/20 0.61
LMNA P02545 1/20 0.53
LRRK2 Q5S007 1/20 0.52
WDR91 A4D1P6 2/20 0.50
PBK Q96KB5 1/20 0.48
PRKDC P78527 1/20 0.47
ALDH1A1 P00352 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HSD17B10 Q99714 2/20 0.47
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
JAK2 O60674 1/20 0.47
JAK1 P23458 1/20 0.47
SYK P43405 1/20 0.47
JAK3 P52333 1/20 0.47
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2183374 0.90 NOTUM (0.75) KMT2AMEN1NOTUMALDH1A1NPSR1
SCHEMBL16695124 0.90 NOTUM (0.75) KMT2AMEN1NOTUMALDH1A1NPSR1
Hydrochloric Acid SCHEMBL30098430 0.89 NOTUM (0.73) KMT2AMEN1NOTUMALDH1A1NPSR1
SCHEMBL613112 0.87 NOTUM (0.81) KMT2AMEN1NOTUMALDH1A1HSD17B10
SCHEMBL4961935 0.87 NOTUM (0.81) KMT2AMEN1NOTUMALDH1A1HSD17B10
SCHEMBL79756 0.86 WDR91 (0.52) KMT2AMEN1NOTUMLMNALRRK2
SCHEMBL2448228 0.84 WDR91 (0.51) KMT2AMEN1NOTUMLMNAWDR91
SCHEMBL2449550 0.84 NOTUM (0.61) KMT2AMEN1NOTUMWDR91PBK
SCHEMBL2451481 0.84 WDR91 (0.66) KMT2AMEN1NOTUMWDR91PBK
SCHEMBL2449229 0.84 NOTUM (0.64) KMT2AMEN1NOTUMLMNAWDR91

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758580-A4 N-SUBSTITUTED PIPERIDINES AND THEIR USE AS PHARMACEUTICALS INCYTE CORP (US) 2008-01-16 EP claimed
EP-1758580-A2 N-SUBSTITUTED PIPERIDINES AND THEIR USE AS PHARMACEUTICALS Incyte Corporation (US) 2007-03-07 EP claimed
WO-2006012226-A2 N-SUBSTITUTED PIPERIDINES AND THEIR USE AS PHARMACEUTICALS INCYTE CORPORATION (US) 2006-02-02 WO claimed
US-12419888-B2 Methods of treating elevated plasma cholesterol INSTITUT DE CARDIOLOGIE DE MONTREAL (CA) 2025-09-23 US disclosed
US-20220296593-A1 METHODS OF TREATING ELEVATED PLASMA CHOLESTEROL INSTITUT DE CARDIOLOGIE DE MONTREAL (CA) 2022-09-22 US disclosed
CN-114746151-A Aryl heterocyclic compounds as Kv1.3 potassium Shaker channel blockers D·E·萧尔研究有限责任公司 2022-07-12 CN disclosed
EP-2362775-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2011-09-07 EP disclosed
WO-2010059658-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-05-27 WO disclosed
CN-1297559-C Fused bicyclic pyrimidine derivatives KYORIN SEIYAKU KK (JP) 2007-01-31 CN disclosed
CN-1620459-A Fused bicyclic pyrimidine derivatives KYORIN SEIYAKU KK (JP) 2005-05-25 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220296593-A1 METHODS OF TREATING ELEVATED PLASMA CHOLESTEROL PCSK9, LDLR, CETP KMT2A 3355/4885MEN1 1446/4885NOTUM 507/4885
US-12419888-B2 Methods of treating elevated plasma cholesterol PCSK9, LDLR, CETP KMT2A 3307/4885MEN1 1583/4885NOTUM 473/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.