SCHEMBL24468617

SCHEMBL24468617

CN(Cc1ccc(C(F)(F)F)cn1)C(=O)c1ccc2nc(N)c3c(c2c1)COC3

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 2/20 0.49
WDR77 Q9BQA1 1/20 0.49
TRPM8 Q7Z2W7 2/20 0.41
ITGB3 P05106 1/20 0.38
ITGAV P06756 1/20 0.38
SCN9A Q15858 4/20 0.38
MCHR1 Q99705 3/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NLRP3 Q96P20 1/20 0.36
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
TACR1 P25103 1/20 0.35
ROCK2 O75116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29685468 1.00 PRMT5 (0.49) PRMT5WDR77TRPM8ITGB3ITGAV
SCHEMBL29685483 1.00 PRMT5 (0.49) PRMT5WDR77TRPM8ITGB3ITGAV
SCHEMBL27181245 0.91 PRMT5 (0.48) PRMT5WDR77TRPM8SCN9AMCHR1
SCHEMBL29685302 0.90 PRMT5 (0.48) PRMT5WDR77TRPM8SCN9AMCHR1
SCHEMBL24468560 0.90 PRMT5 (0.48) PRMT5WDR77TRPM8SCN9AMCHR1
SCHEMBL27472839 0.90 PRMT5 (0.48) PRMT5WDR77TRPM8ITGB3ITGAV
SCHEMBL30971468 0.90 PRMT5 (0.48) PRMT5WDR77TRPM8ITGB3ITGAV
SCHEMBL24468619 0.90 PRMT5 (0.47) PRMT5WDR77TRPM8SCN9AMCHR1
SCHEMBL29685406 0.90 PRMT5 (0.47) PRMT5WDR77TRPM8SCN9AMCHR1
SCHEMBL24468123 0.89 PRMT5 (0.54) PRMT5WDR77TRPM8SCN9AMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116783191-A Tricyclic carboxamide derivatives as PRMT5 inhibitors 美国安进公司 2023-09-19 CN claimed
CN-116783191-A Tricyclic carboxamide derivatives as PRMT5 inhibitors 美国安进公司 2023-09-19 CN disclosed
WO-2022115377-A1 TRICYCLIC CARBOXAMIDE DERIVATIVES AS PRMT5 INHIBITORS AMGEN INC. (US) 2022-06-02 WO disclosed