SCHEMBL244760

SCHEMBL244760

CNC(=O)c1cccc(CCSc2nc(N)c(C#N)c(-c3ccc(OCCO)cc3)c2C#N)c1

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 18/20 0.71
ADORA2B P29275 4/20 0.58
ADORA3 P0DMS8 1/20 0.56
KDM4E B2RXH2 1/20 0.54
MEN1 O00255 1/20 0.54
USP2 O75604 1/20 0.54
ALDH1A1 P00352 1/20 0.54
TP53 P04637 1/20 0.54
MAPT P10636 1/20 0.54
HPGD P15428 1/20 0.54
ALOX15 P16050 1/20 0.54
KMT2A Q03164 1/20 0.54
HSD17B10 Q99714 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL245503 0.93 ADORA1 (0.72) ADORA1ADORA2B
SCHEMBL254320 0.91 ADORA1 (0.70) ADORA1ADORA2BADORA3KDM4EMEN1
SCHEMBL3361524 0.86 ADORA1 (0.65) ADORA1ADORA2BADORA3KDM4EMEN1
SCHEMBL244063 0.85 ADORA1 (0.77) ADORA1ADORA2BKDM4EMEN1USP2
SCHEMBL244025 0.85 ADORA1 (0.70) ADORA1ADORA2B
SCHEMBL12503198 0.83 ADORA1 (0.67) ADORA1ADORA2BKDM4EMEN1USP2
SCHEMBL244759 0.83 ADORA1 (1.00) ADORA1ADORA2BADORA3KDM4EMEN1
SCHEMBL3337662 0.83 ADORA1 (1.00) ADORA1ADORA2BADORA3KDM4EMEN1
SCHEMBL382292 0.82 ADORA1 (0.76) ADORA1ADORA2BADORA3KDM4EMEN1
SCHEMBL244002 0.80 ADORA1 (0.79) ADORA1ADORA2BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588454-A1 SUBSTITUTED DICYANOPYRIDINES AND USE THEREOF Bayer Intellectual Property GmbH (DE) 2013-05-08 EP disclosed
WO-2012000945-A1 SUBSTITUTED DICYANOPYRIDINES AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-01-05 WO disclosed