SCHEMBL2447664

SCHEMBL2447664

COc1ccc2ncc3c(c2n1)C(CN1CCC(NCc2ccc4c(n2)NC(=O)CO4)C(CO)C1)CO3

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 17/20 0.57
KCNQ1 P51787 1/20 0.51
CACNA1C Q13936 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2447658 1.00 KCNH2 (0.57) KCNH2KCNQ1CACNA1C
SCHEMBL2448181 0.92 KCNH2 (0.62) KCNH2KCNQ1CACNA1C
SCHEMBL2448185 0.92 KCNH2 (0.62) KCNH2KCNQ1CACNA1C
SCHEMBL2445323 0.89 KCNH2 (0.46) KCNH2
SCHEMBL2445325 0.89 KCNH2 (0.46) KCNH2
SCHEMBL1074325 0.89 KCNH2 (0.69) KCNH2KCNQ1CACNA1C
SCHEMBL1267277 0.86 KCNH2 (0.56) KCNH2KCNQ1CACNA1C
SCHEMBL1267369 0.85 KCNH2 (0.53) KCNH2KCNQ1CACNA1C
SCHEMBL1266381 0.85 KCNH2 (0.53) KCNH2KCNQ1CACNA1C
SCHEMBL1267287 0.83 KCNH2 (0.59) KCNH2KCNQ1CACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012961-B2 Tricyclic antibiotics ACTELION PHARMACEUTICAL LTD. (CH) 2011-09-06 US disclosed