SCHEMBL24520064

SCHEMBL24520064

Cc1ccc(-c2ccc3ncc(C#Cc4cc(N)nc5[nH]ccc45)n3c2)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 1/20 0.34
RPS6KA3 P51812 1/20 0.33
PRKCA P17252 1/20 0.33
PRKCI P41743 1/20 0.33
PRKCE Q02156 1/20 0.33
TGFBR1 P36897 5/20 0.32
NTRK1 P04629 5/20 0.32
NTRK3 Q16288 5/20 0.32
NTRK2 Q16620 5/20 0.32
KDM4E B2RXH2 2/20 0.31
NPC1 O15118 2/20 0.31
ALDH1A1 P00352 2/20 0.31
RAB9A P51151 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
NPSR1 Q6W5P4 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
LMNA P02545 1/20 0.31
PIK3CA P42336 1/20 0.30
PRMT5 O14744 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16621078 0.89 PIK3CA (0.32) CSNK1DPRKCAPRKCIPRKCETGFBR1
SCHEMBL24520056 0.88 PIK3CA (0.31) CSNK1DPIK3CA
SCHEMBL16620670 0.81 MKNK1 (0.49) PIK3CA
SCHEMBL16620931 0.81 MKNK1 (0.49) NTRK3PIK3CA
SCHEMBL29756308 0.81 MKNK1 (0.49) NTRK3PIK3CA
SCHEMBL17969545 0.73 PRKCI (0.37) CSNK1DRPS6KA3PRKCAPRKCIPRKCE
SCHEMBL24520037 0.71 PRKCI (0.36) RPS6KA3PRKCAPRKCIPRKCENTRK3
SCHEMBL24520074 0.71 CSNK1D (0.35) CSNK1DTGFBR1PIK3CAPRMT5WDR77
SCHEMBL18012832 0.71 MKNK1 (0.51) NTRK3
SCHEMBL16626035 0.65 MKNK1 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052501-B1 BICYCLIC ALKYNE DERIVATIVES AND USES THEREOF AGENCY SCIENCE TECH & RES (SG) 2022-06-22 EP disclosed