SCHEMBL2452544

SCHEMBL2452544

CCCCCC1CCC(Oc2ccc3cc(C(C)(C)N)ccc3c2)CC1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.35
ROCK1 Q13464 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
MAOA P21397 2/20 0.32
MAOB P27338 2/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C8 P10632 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
S1PR3 Q99500 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
PTPN1 P18031 1/20 0.32
IKBKB O14920 1/20 0.32
PARP1 P09874 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2454249 0.91 KCNH2 (0.36) KCNH2ROCK1MAOAMAOBCYP2C9
SCHEMBL2450020 0.91 KCNH2 (0.40) KCNH2ROCK1L3MBTL1MAOAMAOB
SCHEMBL2450402 0.91 KCNH2 (0.40) KCNH2ROCK1L3MBTL1MAOAMAOB
SCHEMBL2450023 0.91 KCNH2 (0.40) KCNH2ROCK1L3MBTL1MAOAMAOB
SCHEMBL2451700 0.91 KCNH2 (0.40) KCNH2ROCK1L3MBTL1MAOAMAOB
SCHEMBL2778723 0.87 KCNH2 (0.40) KCNH2ROCK1L3MBTL1MAOAMAOB
SCHEMBL2446408 0.87 KCNH2 (0.40) KCNH2ROCK1L3MBTL1MAOAMAOB
SCHEMBL2777420 0.87 KCNH2 (0.40) KCNH2ROCK1L3MBTL1MAOAMAOB
SCHEMBL16457167 0.87 KCNH2 (0.34) KCNH2ROCK1L3MBTL1MAOAMAOB
SCHEMBL2777477 0.87 KCNH2 (0.40) KCNH2ROCK1L3MBTL1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364088-A1 BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS Biogen Idec MA Inc. (US) 2011-09-14 EP claimed
WO-2010051030-A1 BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS BIOGEN IDEC MA INC. (US) 2010-05-06 WO claimed
EP-2364088-A1 BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS Biogen Idec MA Inc. (US) 2011-09-14 EP disclosed
WO-2010051030-A1 BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS BIOGEN IDEC MA INC. (US) 2010-05-06 WO disclosed