SCHEMBL24528060

SCHEMBL24528060

c1ccc(-c2ccc3c(c2)c2cc(-c4ccccc4)ccc2n3-c2cc3c4ccncc4n4c5cnccc5c(c2)c34)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 3/20 0.36
MKNK1 Q9BUB5 1/20 0.35
NR3C1 P04150 1/20 0.35
PIK3CA P42336 1/20 0.35
MAPK10 P53779 1/20 0.34
KCNH2 Q12809 2/20 0.34
GSK3B P49841 1/20 0.34
NPY5R Q15761 1/20 0.33
DHODH Q02127 1/20 0.33
MEN1 O00255 1/20 0.33
HSP90AA1 P07900 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ATM Q13315 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CDK4 P11802 1/20 0.32
CDK6 Q00534 1/20 0.32
CYP1A2 P05177 1/20 0.32
METAP2 P50579 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528000 0.90 KDM4E (0.44) DYRK1AKCNH2GSK3BNPY5RMEN1
SCHEMBL24527994 0.89 KDM4E (0.45) DYRK1AKCNH2GSK3BNPY5RMEN1
SCHEMBL24528219 0.86 DYRK1A (0.40) DYRK1AMKNK1PIK3CAMAPK10KCNH2
SCHEMBL24528193 0.86 DYRK1A (0.40) DYRK1AMKNK1PIK3CAMAPK10KCNH2
SCHEMBL17704962 0.86 KDM4E (0.40) DYRK1AMKNK1NR3C1KCNH2GSK3B
SCHEMBL15945736 0.85 CDK4 (0.42) DYRK1AMKNK1NR3C1PIK3CAMAPK10
SCHEMBL11965527 0.85 CDK4 (0.42) DYRK1AMKNK1NR3C1PIK3CAMAPK10
SCHEMBL25946458 0.85 KDM4E (0.44) DYRK1AMKNK1PIK3CAMAPK10KCNH2
SCHEMBL17704977 0.85 KDM4E (0.44) DYRK1AKCNH2GSK3BNPY5RKDM4E
SCHEMBL17265101 0.85 KDM4E (0.44) DYRK1AKCNH2GSK3BNPY5RKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129113-A1 NITROGENOUS HETEROAROMATIC COMPOUNDS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2022-06-23 WO disclosed