SCHEMBL24534091

SCHEMBL24534091

O=CNc1cc(C(F)(F)F)c(C=O)cn1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 4/20 0.35
AR P10275 1/20 0.33
KIF11 P52732 1/20 0.31
ASPH Q12797 1/20 0.30
CCNE2 O96020 1/20 0.30
CDK4 P11802 1/20 0.30
CCND1 P24385 1/20 0.30
CCNE1 P24864 1/20 0.30
CDK2 P24941 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22509078 0.81 TEK (0.36) AR
SCHEMBL27743601 0.77 ERN1 (0.37) ERN1KIF11ASPH
SCHEMBL29728357 0.75 KDR (0.42) AR
SCHEMBL23140058 0.75 AAK1 (0.40)
SCHEMBL16611723 0.75 KDR (0.42) AR
SCHEMBL3783458 0.75 KCNQ3 (0.37) ERN1KIF11ASPH
SCHEMBL2439088 0.75 ALOX5AP (0.39) ERN1
SCHEMBL30445332 0.75 KCNQ3 (0.37) ERN1KIF11ASPH
SCHEMBL4649615 0.71 CNR2 (0.53)
SCHEMBL3779382 0.71 MAPT (0.45) ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022128850-A1 NOVEL ISOQUINOLINE DERIVATIVES AND PHARMACEUTICAL COPOSITIONS THEREOF FOR THE TREATMENT OF DISEASES GALAPAGOS NV (BE) 2022-06-23 WO disclosed