SCHEMBL24543293

SCHEMBL24543293

COC(=O)C12CCCN1C[C@H](F)C2

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 2/20 0.33
OPRD1 P41143 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
OPRM1 P35372 1/20 0.32
PPIA P62937 1/20 0.31
ALDH1A1 P00352 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30885335 1.00 OPRL1 (0.33) OPRL1OPRD1NPSR1OPRM1PPIA
SCHEMBL26893877 1.00 OPRL1 (0.33) OPRL1OPRD1NPSR1OPRM1PPIA
SCHEMBL29940079 1.00 OPRL1 (0.33) OPRL1OPRD1NPSR1OPRM1PPIA
SCHEMBL29940065 1.00 OPRL1 (0.33) OPRL1OPRD1NPSR1OPRM1PPIA
SCHEMBL29851149 0.93 NPSR1 (0.31) NPSR1
SCHEMBL24649055 0.93 NPSR1 (0.31) NPSR1
SCHEMBL26893933 0.84 OPRL1 (0.33) OPRL1OPRD1NPSR1OPRM1PPIA
SCHEMBL31442177 0.84 OPRL1 (0.33) OPRL1OPRD1NPSR1OPRM1PPIA
SCHEMBL30922808 0.84 OPRL1 (0.33) OPRL1OPRD1NPSR1OPRM1PPIA
SCHEMBL30709846 0.83 TSHR (0.32) NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250059205-A1 Heterocyclic Compounds and Methods of Use AMGEN INC. (US) 2025-02-20 US disclosed
US-20250059179-A1 Heterocyclic Compounds and Methods of Use AMGEN INC. (US) 2025-02-20 US disclosed
EP-4329888-A1 2-AMINOBENZOTHIAZOLE COMPOUNDS AND METHODS OF USE THEREOF Amgen Inc. (US) 2024-03-06 EP disclosed
US-11548888-B2 KRas G12C inhibitors Mirati Therapeutics, Inc. (US) 2023-01-10 US disclosed
EP-4087573-A1 KRAS G12C INHIBITORS Mirati Therapeutics, Inc. (US) 2022-11-16 EP disclosed
WO-2022232332-A1 2-AMINOBENZOTHIAZOLE COMPOUNDS AND METHODS OF USE THEREOF AMGEN INC. (US) 2022-11-03 WO disclosed
WO-2022127827-A1 KRASG12C PROTEIN MUTATION INHIBITOR AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 上海维申医药有限公司 2022-06-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250059179-A1 Heterocyclic Compounds and Methods of Use KRAS, NRAS, HRAS OPRL1 4567/4885OPRD1 2932/4885NPSR1 4800/4885
US-20250059205-A1 Heterocyclic Compounds and Methods of Use KRAS, NRAS, HRAS OPRL1 4567/4885OPRD1 2932/4885NPSR1 4800/4885
US-11548888-B2 KRas G12C inhibitors KRAS, NRAS, HRAS OPRL1 4628/4885OPRD1 4708/4885NPSR1 4791/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.