SCHEMBL24558142

SCHEMBL24558142

COc1cc(-c2c(O)cccc2F)c(Cl)c2c1C(=O)N1CCN(C(=O)OC(C)(C)C)C[C@@H]1CO2

nearest known ligand 0.49

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KRAS P01116 19/20 0.49
USP30 Q70CQ3 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29693198 1.00 KRAS (0.49) KRASUSP30
SCHEMBL24558433 0.91 KRAS (0.54) KRASUSP30
SCHEMBL28673539 0.90 KRAS (0.52) KRAS
SCHEMBL29693150 0.86 KRAS (0.54) KRAS
SCHEMBL30240561 0.84 KRAS (0.42) KRASUSP30
SCHEMBL24069449 0.84 KRAS (0.42) KRASUSP30
SCHEMBL25698396 0.84 KRAS (0.44) KRASUSP30
SCHEMBL24069210 0.83 KRAS (0.44) KRASUSP30
SCHEMBL30240226 0.83 KRAS (0.44) KRASUSP30
SCHEMBL30240406 0.83 KRAS (0.44) KRASUSP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3935060-B1 FUSED TRICYCLIC COMPOUNDS USEFUL AS ANTICANCER AGENTS ASTRAZENECA AB (SE) 2023-11-15 EP disclosed
US-20220204527-A1 FUSED TRICYCLIC COMPOUNDS USEFUL AS ANTICANCER AGENTS ASTRAZENECA UK LIMITED (GB) 2022-06-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220204527-A1 FUSED TRICYCLIC COMPOUNDS USEFUL AS ANTICANCER AGENTS MCL1, TP53, CCNA2 KRAS 89/4885USP30 4265/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.