SCHEMBL2458459

SCHEMBL2458459

COc1ccc(C(=O)O)c2nc(C3CCCC3)[nH]c12

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.64
PDE4B Q07343 3/20 0.64
PDE4C Q08493 3/20 0.64
PDE4D Q08499 3/20 0.64
PBK Q96KB5 11/20 0.44
ADORA3 P0DMS8 2/20 0.43
ADORA1 P30542 2/20 0.43
GSK3B P49841 1/20 0.43
PARP1 P09874 1/20 0.40
HTR2B P41595 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1581071 0.95 PDE4A (0.63) PDE4APDE4BPDE4CPDE4DPBK
SCHEMBL1554160 0.90 PDE4A (0.56) PDE4APDE4BPDE4CPDE4DPBK
Hydrochloric Acid SCHEMBL8576071 0.89 PDE4A (0.55) PDE4APDE4BPDE4CPDE4DPBK
SCHEMBL1581014 0.89 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DPBK
SCHEMBL1552957 0.85 PDE4D (0.54) PDE4APDE4BPDE4CPDE4DPBK
Hydrochloric Acid SCHEMBL8568573 0.84 PDE4D (0.53) PDE4APDE4BPDE4CPDE4DPBK
SCHEMBL2318486 0.84 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DPBK
SCHEMBL8571281 0.82 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DPBK
SCHEMBL1581259 0.82 PBK (0.61) PDE4APDE4BPDE4CPDE4DPBK
SCHEMBL1554161 0.81 PDE4A (0.58) PDE4APDE4BPDE4CPDE4DPBK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364087-A1 7-HYDROXY-BENZOIMIDAZOLE-4-YL-METHANONE DERIVATIVES AND PBK INHIBITORS CONTAINING THE SAME Oncotherapy Science, Inc. (JP) 2011-09-14 EP disclosed
WO-2010051085-A1 7-HYDROXY-BENZOIMIDAZOLE-4-YL-METHANONE DERIVATIVES AND PBK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2010-05-06 WO disclosed