SCHEMBL24586249

SCHEMBL24586249

Cc1cc(CC(=O)Nc2cc(C3CC[C@@H](OC(=O)NC45CC(C4)C5)C3)[nH]n2)on1

nearest known ligand 0.81

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 20/20 0.81
CCNE1 P24864 19/20 0.81
GSK3B P49841 15/20 0.81
CDK1 P06493 1/20 0.81
CDK4 P11802 1/20 0.81
CCNA2 P20248 1/20 0.81
CCND1 P24385 1/20 0.81
CDK9 P50750 1/20 0.81
CDK6 Q00534 1/20 0.81

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24586157 1.00 CDK2 (0.81) CDK2CCNE1GSK3BCDK1CDK4
SCHEMBL24586153 1.00 CDK2 (0.81) CDK2CCNE1GSK3BCDK1CDK4
SCHEMBL24585229 1.00 CDK2 (0.81) CDK2CCNE1GSK3BCDK1CDK4
SCHEMBL24586251 1.00 CDK2 (0.81) CDK2CCNE1GSK3BCDK1CDK4
SCHEMBL24586144 1.00 CDK2 (0.81) CDK2CCNE1GSK3BCDK1CDK4
SCHEMBL26041769 0.89 CDK2 (1.00) CDK2CCNE1GSK3BCDK1CDK4
SCHEMBL22310620 0.89 CDK2 (1.00) CDK2CCNE1GSK3BCDK1CDK4
SCHEMBL22311799 0.89 CDK2 (1.00) CDK2CCNE1GSK3BCDK1CDK4
SCHEMBL22287121 0.86 CDK2 (1.00) CDK2CCNE1GSK3BCDK1CDK4
SCHEMBL22311433 0.86 CDK2 (1.00) CDK2CCNE1GSK3BCDK1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022135442-A1 CDK2 INHIBITOR AND PREPARATION METHOD THEREFOR 上海拓界生物医药科技有限公司 2022-06-30 WO disclosed