SCHEMBL24601694

SCHEMBL24601694

O=C(/C=C/C=C/c1ccc2c(c1)OCO2)OC(=O)/C=C/C=C/c1ccc2c(c1)OCO2

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.74
HSD17B10 Q99714 3/20 0.74
CYP1A2 P05177 2/20 0.74
HDAC6 Q9UBN7 2/20 0.68
MAOA P21397 2/20 0.67
KDM4E B2RXH2 3/20 0.63
ALDH1A1 P00352 3/20 0.63
GABRA1 P14867 4/20 0.62
GABRB2 P47870 4/20 0.62
TRPV1 Q8NER1 3/20 0.62
CYP3A4 P08684 2/20 0.62
HPGD P15428 2/20 0.62
SMN1; SMN2 Q16637 2/20 0.62
NPC1 O15118 1/20 0.62
CTSD P07339 1/20 0.62
ABCB1 P08183 1/20 0.62
ALOX5 P09917 1/20 0.62
MAPK1 P28482 1/20 0.62
RAB9A P51151 1/20 0.62
DHODH Q02127 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3804124 0.90 MAOB (0.72) MAOBHSD17B10CYP1A2HDAC6MAOA
Methyl Piperate SCHEMBL3244271 0.89 KDM4E (0.82) MAOBHSD17B10CYP1A2HDAC6MAOA
Methyl Piperate SCHEMBL2328493 0.89 KDM4E (0.82) MAOBHSD17B10CYP1A2HDAC6MAOA
SCHEMBL22128483 0.86 MAOB (0.67) MAOBHSD17B10CYP1A2HDAC6MAOA
SCHEMBL29251152 0.86 MAOB (0.67) MAOBHSD17B10CYP1A2HDAC6MAOA
SCHEMBL10733556 0.85 MAOB (0.71) MAOBHSD17B10CYP1A2HDAC6MAOA
SCHEMBL10733568 0.85 MAOB (0.71) MAOBHSD17B10CYP1A2HDAC6MAOA
SCHEMBL17340491 0.85 MAOB (0.66) MAOBHSD17B10CYP1A2HDAC6MAOA
SCHEMBL28042612 0.85 MAOB (0.66) MAOBHSD17B10CYP1A2HDAC6MAOA
Piperic Acid SCHEMBL11460092 0.85 HSD17B10 (1.00) MAOBHSD17B10CYP1A2HDAC6MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022146980-A1 COMPOSITIONS AND METHODS FOR INHIBITING FIBROSIS, INFLAMMATION AND CANCER GEORGIA TECH RESEARCH CORPORATION (US) 2022-07-07 WO disclosed