SCHEMBL2460932

SCHEMBL2460932

O=CCN1CCCC(c2cccnc2Oc2ccc(Nc3nc4ccccc4s3)cc2)C1

nearest known ligand 0.77

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 20/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2461647 1.00 PDE10A (0.77) PDE10A
SCHEMBL2455427 0.91 PDE10A (0.73) PDE10A
SCHEMBL2460350 0.87 PDE10A (1.00) PDE10A
SCHEMBL3317103 0.87 PDE10A (1.00) PDE10A
SCHEMBL2461642 0.87 PDE10A (1.00) PDE10A
SCHEMBL13361556 0.84 PDE10A (0.84) PDE10A
SCHEMBL2462238 0.83 PDE10A (0.90) PDE10A
SCHEMBL2366922 0.83 PDE10A (0.59) PDE10A
SCHEMBL2455900 0.81 PDE10A (1.00) PDE10A
SCHEMBL13332645 0.81 PDE10A (1.00) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364306-A1 Pyridine and pyrimidine derivatives as phosphodiesterase 10 inhibitors Amgen Inc. (US) 2011-09-14 EP disclosed
WO-2010057126-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AS PHOSPHODIESTERASE 10 INHIBITORS AMGEN INC. (US) 2010-05-20 WO disclosed