SCHEMBL24626403

SCHEMBL24626403

Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1C#Cc1cnc(N)c(C)c1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 10/20 0.83
KDR P35968 8/20 0.83
TEK Q02763 7/20 0.83
KIT P10721 6/20 0.69
DDR1 Q08345 1/20 0.69
DDR2 Q16832 1/20 0.69
CSF1R P07333 3/20 0.67
SRC P12931 4/20 0.62
ABL1 P00519 3/20 0.61
MAPK14 Q16539 4/20 0.59
BCR P11274 1/20 0.57
KDM4E B2RXH2 1/20 0.57
MAPT P10636 1/20 0.57
FYN P06241 1/20 0.56
YES1 P07947 1/20 0.56
LYN P07948 1/20 0.56
HCK P08631 1/20 0.56
FGR P09769 1/20 0.56
CSK P41240 1/20 0.56
BLK P51451 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2969534 0.91 LCK (1.00) LCKKDRTEKKITDDR1
SCHEMBL3430966 0.90 LCK (0.75) LCKKDRTEKKITDDR1
SCHEMBL2974278 0.89 LCK (1.00) LCKKDRTEKKITDDR1
SCHEMBL2975413 0.85 LCK (1.00) LCKKDRTEKKITDDR1
SCHEMBL14953284 0.85 LCK (0.77) LCKKDRTEKKITDDR1
SCHEMBL29515236 0.85 LCK (0.77) LCKKDRTEKKITDDR1
SCHEMBL3586277 0.84 TEK (0.77) LCKKDRTEKKITDDR1
SCHEMBL3574810 0.84 LCK (1.00) LCKKDRTEKKITDDR1
SCHEMBL2976092 0.83 LCK (0.86) LCKKDRTEKKITDDR1
SCHEMBL17325058 0.83 LCK (0.73) LCKKDRTEKKITDDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022149855-A1 HETEROARYL-ETHYNYL DERIVATIVE COMPOUND AND USE THEREOF 주식회사 비투에스바이오 2022-07-14 WO disclosed