SCHEMBL24640437

SCHEMBL24640437

CN1CCN2c3ncc(C(F)(F)F)cc3N[C@H]2C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TIPARP Q7Z3E1 2/20 0.44
SMN1; SMN2 Q16637 5/20 0.40
LMNA P02545 2/20 0.40
POLB P06746 1/20 0.36
HRH4 Q9H3N8 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CXCR3 P49682 2/20 0.33
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
KCNH2 Q12809 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
MDM2 Q00987 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24639862 0.84 TIPARP (0.46) TIPARPSMN1; SMN2POLBHRH3CXCR3
SCHEMBL26958125 0.79 TIPARP (0.47) TIPARPSMN1; SMN2LMNAPOLBHRH4
SCHEMBL31244646 0.79 GAA (0.41) TIPARPSMN1; SMN2LMNAPOLBALDH1A1
SCHEMBL31244762 0.78 HTR2C (0.40) TIPARPPOLBHTR2AHTR2CHTR2B
SCHEMBL31244702 0.78 HTR2C (0.40) TIPARPPOLBHTR2AHTR2CHTR2B
SCHEMBL31244748 0.78 HTR2C (0.40) TIPARPPOLBHTR2AHTR2CHTR2B
SCHEMBL24639905 0.78 TIPARP (0.49) TIPARPSMN1; SMN2LMNAMDM2NPC1
SCHEMBL24639557 0.78 TIPARP (0.49) TIPARPSMN1; SMN2LMNAMDM2NPC1
SCHEMBL24639530 0.78 TIPARP (0.49) TIPARPSMN1; SMN2LMNAMDM2NPC1
SCHEMBL26958206 0.74 SMN1; SMN2 (0.40) SMN1; SMN2LMNAPOLBHRH4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022170974-A1 TRICYCLIC DERIVATIVES USEFUL AS PARP7 INHIBITORS JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2022-08-18 WO disclosed