SCHEMBL24655243

SCHEMBL24655243

CC1(C)c2ccccc2-c2ccc(N(c3ccc(-c4ccc5c(ccc6ccc7ccccc7c65)c4)cc3)c3cccc(-c4ccccc4)c3)cc21

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.32
CCND1 P24385 1/20 0.32
PDK2 Q15119 3/20 0.32
HSD17B1 P14061 1/20 0.32
HSD17B2 P37059 1/20 0.32
CYP1A1 P04798 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP1B1 Q16678 1/20 0.31
CA12 O43570 2/20 0.30
CA1 P00915 2/20 0.30
CA2 P00918 2/20 0.30
CA9 Q16790 2/20 0.30
SLC6A9 P48067 1/20 0.30
CHRNA1 P02708 1/20 0.30
CHRNG P07510 1/20 0.30
CHRNB1 P11230 1/20 0.30
CHRNB2 P17787 1/20 0.30
SLC6A2 P23975 1/20 0.30
CHRNB4 P30926 1/20 0.30
SLC6A4 P31645 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24655247 0.97 CHRNA1 (0.33) HSD17B1HSD17B2CYP1A1CYP1A2CYP1B1
SCHEMBL24655241 0.97 PDK2 (0.33) PDK2HSD17B1HSD17B2
SCHEMBL24655253 0.97 PDK2 (0.33) PDK2
SCHEMBL24655246 0.96 CHRNA1 (0.34) CYP1A1CYP1A2CYP1B1CA12CA1
SCHEMBL24657952 0.96 CDK4 (0.33) CDK4CCND1PDK2CYP1A1CYP1A2
SCHEMBL24657698 0.95 CA12 (0.34) CDK4CCND1PDK2CYP1A1CYP1A2
SCHEMBL24658059 0.95 CDK4 (0.32) CDK4CCND1PDK2CA12CA1
SCHEMBL24655252 0.95 PDK2 (0.31) PDK2CA12CA1CA2CA9
SCHEMBL24657959 0.94 CHRNA1 (0.34) PDK2HSD17B1HSD17B2CYP1A1CYP1A2
SCHEMBL24655254 0.94 CDK4 (0.32) CDK4CCND1HSD17B1HSD17B2CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4243100-A1 ORGANIC LIGHT-EMITTING DEVICE Lg Chem, Ltd. (KR) 2023-09-13 EP disclosed
WO-2022177374-A1 ORGANIC LIGHT-EMITTING DEVICE 주식회사 엘지화학 2022-08-25 WO disclosed