SCHEMBL24664327

SCHEMBL24664327

Cc1cnc(Nc2ccc(N)c(F)c2)nc1-c1cnn(C(C)C)c1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 20/20 0.61
TYK2 P29597 9/20 0.61
JAK1 P23458 8/20 0.61
JAK3 P52333 8/20 0.61
FLT3 P36888 15/20 0.59
CYP1A2 P05177 1/20 0.58
LCK P06239 1/20 0.58
LYN P07948 1/20 0.58
CYP2C9 P11712 1/20 0.58
CDK4 P11802 1/20 0.58
FLT1 P17948 1/20 0.58
CCND3 P30281 1/20 0.58
CYP2C19 P33261 1/20 0.58
FLT4 P35916 1/20 0.58
CDK6 Q00534 1/20 0.58
KCNH2 Q12809 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29608214 0.84 JAK2 (0.64) JAK2TYK2JAK1JAK3FLT3
SCHEMBL29527869 0.83 JAK2 (0.65) JAK2TYK2JAK1JAK3FLT3
SCHEMBL29608225 0.82 JAK2 (0.75) JAK2TYK2JAK1JAK3FLT3
SCHEMBL24664433 0.82 JAK2 (0.75) JAK2TYK2JAK1JAK3FLT3
SCHEMBL22852642 0.81 JAK2 (0.69) JAK2TYK2JAK1JAK3FLT3
SCHEMBL24664434 0.80 JAK2 (0.71) JAK2TYK2JAK1JAK3FLT3
SCHEMBL29607219 0.80 JAK2 (0.71) JAK2TYK2JAK1JAK3FLT3
Hydrochloric Acid SCHEMBL31460911 0.79 JAK2 (0.69) JAK2TYK2JAK1JAK3FLT3
SCHEMBL29425676 0.79 JAK2 (0.58) JAK2TYK2JAK1JAK3FLT3
SCHEMBL29741634 0.79 JAK2 (0.68) JAK2TYK2JAK1JAK3FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114423750-B 2, 4-Disubstituted pyrimidine derivative, preparation method and application thereof 成都赜灵生物医药科技有限公司 2024-04-19 CN disclosed
US-20220298140-A1 2,4-DISUBSTITUTED PYRIMIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF CHENGDU ZENITAR BIOMEDICAL TECHNOLOGY CO., LTD. (CN) 2022-09-22 US disclosed
CN-114423750-A 2, 4-disubstituted pyrimidine derivative and preparation method and application thereof 成都赜灵生物医药科技有限公司 2022-04-29 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220298140-A1 2,4-DISUBSTITUTED PYRIMIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF JAK2, FLT3, JAK1 JAK2 1/4885TYK2 15/4885JAK1 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.