SCHEMBL2466686

SCHEMBL2466686

Cc1c(C(F)(F)F)ccc2c1nc(N1CCNCC1)c1nnnn12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.43
EPHX2 P34913 1/20 0.41
MAPT P10636 6/20 0.41
TP53 P04637 2/20 0.40
KDM4E B2RXH2 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ADRB2 P07550 1/20 0.39
TSHR P16473 2/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
USP2 O75604 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
HRH4 Q9H3N8 3/20 0.38
HRH3 Q9Y5N1 2/20 0.38
HBB P68871 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2534943 0.80 POLB (0.48) POLBMAPTTP53KDM4EMEN1
SCHEMBL462636 0.76 HTR1D (0.59) POLBMAPTTP53KDM4EMEN1
SCHEMBL438686 0.76 TSHR (0.46) POLBEPHX2MAPTTP53KDM4E
SCHEMBL440930 0.76 TSHR (0.46) POLBEPHX2MAPTTP53KDM4E
Hydrochloric Acid SCHEMBL442488 0.76 HTR1D (0.58) POLBMAPTTP53KDM4EMEN1
SCHEMBL442492 0.76 POLB (0.41) POLBEPHX2MAPTTP53KDM4E
SCHEMBL462757 0.76 POLB (0.43) POLBMAPTTP53KDM4EMEN1
SCHEMBL406769 0.75 MAPT (0.49) POLBMAPTTP53KDM4EMEN1
Hydrochloric Acid SCHEMBL438242 0.75 TSHR (0.45) POLBEPHX2MAPTTP53KDM4E
SCHEMBL12224913 0.75 POLB (0.43) POLBMAPTTP53KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011112731-A2 HETEROCYCLIC INHIBITORS OF HISTAMINE RECEPTORS FOR THE TREATMENT OF DISEASE KALYPSYS, INC. (US) 2011-09-15 WO disclosed