SCHEMBL24669271

SCHEMBL24669271

CC(C)(C)OC(=O)N1CC=C(c2ccc(C(=O)Nc3ccc(C4=CCN(C(=O)OC(C)(C)C)CC4)c(F)c3)o2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.46
PDK4 Q16654 1/20 0.44
JAK1 P23458 1/20 0.43
GRM5 P41594 5/20 0.42
GRM1 Q13255 5/20 0.42
WNT3A P56704 1/20 0.42
WDR5 P61964 2/20 0.42
HTR6 P50406 1/20 0.42
SCN9A Q15858 1/20 0.41
MAPKAPK2 P49137 1/20 0.40
CDK9 P50750 3/20 0.40
CCNT1 O60563 1/20 0.40
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB1 P18505 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803539 1.00 NAMPT (0.46) NAMPTPDK4JAK1GRM5GRM1
SCHEMBL24670598 0.90 PDK4 (0.39) NAMPTPDK4JAK1GRM5GRM1
SCHEMBL29803459 0.86 MAPKAPK2 (0.36) NAMPTPDK4JAK1WNT3AWDR5
SCHEMBL29803696 0.85 NAMPT (0.52) NAMPTPDK4JAK1GRM5GRM1
SCHEMBL24669339 0.85 NAMPT (0.52) NAMPTPDK4JAK1GRM5GRM1
SCHEMBL24669868 0.85 NAMPT (0.49) NAMPTPDK4JAK1GRM5GRM1
SCHEMBL29803286 0.85 NAMPT (0.49) NAMPTPDK4JAK1GRM5GRM1
SCHEMBL24669930 0.84 MAPKAPK2 (0.41) MAPKAPK2
SCHEMBL29803008 0.84 MAPKAPK2 (0.41) MAPKAPK2
SCHEMBL24670946 0.82 NAMPT (0.49) NAMPTPDK4JAK1GRM5GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed