SCHEMBL24669352

SCHEMBL24669352

Cc1cc(C2=CCN(C(=O)OC(C)(C)C)CC2)ccc1NC(=O)c1ccc(C2=CCN(C(=O)OC(C)(C)C)CC2)cc1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.53
CDK7 P50613 1/20 0.46
CDK13 Q14004 1/20 0.46
CDK12 Q9NYV4 1/20 0.46
GRM1 Q13255 7/20 0.45
GRM5 P41594 6/20 0.45
TP53 P04637 2/20 0.45
MAPT P10636 2/20 0.45
PDK4 Q16654 1/20 0.45
WNT3A P56704 1/20 0.44
SOS1 Q07889 1/20 0.43
JAK1 P23458 1/20 0.43
SCN9A Q15858 1/20 0.42
GAA P10253 1/20 0.42
WDR5 P61964 1/20 0.42
CCNT1 O60563 1/20 0.42
CDK9 P50750 1/20 0.42
LIPC P11150 1/20 0.42
LIPG Q9Y5X9 1/20 0.42
KIT P10721 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803414 1.00 NAMPT (0.53) NAMPTCDK7CDK13CDK12GRM1
SCHEMBL24669373 0.91 SOS1 (0.49) NAMPTCDK7CDK13CDK12GRM1
SCHEMBL29803317 0.89 NAMPT (0.47) NAMPTCDK7CDK13CDK12GRM1
SCHEMBL24670773 0.89 NAMPT (0.47) NAMPTCDK7CDK13CDK12GRM1
SCHEMBL24670904 0.88 NAMPT (0.47) NAMPTCDK7CDK13CDK12GRM1
SCHEMBL29803647 0.88 NAMPT (0.47) NAMPTCDK7CDK13CDK12GRM1
SCHEMBL29802842 0.88 NAMPT (0.52) NAMPTCDK7CDK13CDK12GRM1
SCHEMBL24669309 0.88 NAMPT (0.52) NAMPTCDK7CDK13CDK12GRM1
SCHEMBL24892052 0.86 NAMPT (0.61) NAMPTCDK7CDK13CDK12GRM1
SCHEMBL29803738 0.86 NAMPT (0.54) NAMPTCDK7CDK13CDK12GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed