SCHEMBL24670014

SCHEMBL24670014

CC(C)(C)OC(=O)NCc1ccc(NC(=O)c2ccc(Br)c(F)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.55
HDAC1 Q13547 4/20 0.50
HDAC6 Q9UBN7 1/20 0.50
MAPT P10636 4/20 0.48
TDP1 Q9NUW8 3/20 0.48
FPR3 P25089 1/20 0.46
FPR2 P25090 1/20 0.46
NPSR1 Q6W5P4 2/20 0.45
XBP1 P17861 1/20 0.45
GPR55 Q9Y2T6 1/20 0.45
PPARG P37231 1/20 0.45
MAOB P27338 1/20 0.44
TP53 P04637 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
EPHX2 P34913 2/20 0.42
NR1H4 Q96RI1 2/20 0.42
STAT3 P40763 2/20 0.42
CTNNB1 P35222 1/20 0.42
TCF7L2 Q9NQB0 1/20 0.42
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803661 0.94 NAMPT (0.58) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL24669207 0.94 NAMPT (0.58) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL29803548 0.89 NAMPT (0.53) NAMPTMAPTMAOBTP53NR1H4
SCHEMBL24669863 0.89 NAMPT (0.53) NAMPTMAPTMAOBTP53NR1H4
SCHEMBL30182179 0.88 NAMPT (0.56) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL30182282 0.88 NAMPT (0.52) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL24891826 0.85 NAMPT (0.58) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL23899245 0.85 NAMPT (0.72) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL24670224 0.84 NAMPT (0.65) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL24891860 0.84 NAMPT (0.65) NAMPTHDAC1HDAC6MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed