SCHEMBL24670097

SCHEMBL24670097

CSc1ncc(CO)c(NC(C)S(N)(=O)=O)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.42
CDK1 P06493 3/20 0.33
KDR P35968 3/20 0.33
CA2 P00918 3/20 0.33
CDK4 P11802 2/20 0.33
CDK2 P24941 2/20 0.33
CDK7 P50613 2/20 0.33
CDK9 P50750 2/20 0.33
CCNT1 O60563 1/20 0.33
CCND1 P24385 1/20 0.33
CCNH P51946 1/20 0.33
ALDH1A1 P00352 2/20 0.33
CCNB1 P14635 1/20 0.33
CCNE1 P24864 1/20 0.33
MAPT P10636 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
SYK P43405 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
THRB P10828 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1521541 0.82 HTT (0.48) HTTALDH1A1MAPTSMN1; SMN2SYK
SCHEMBL23142016 0.80 HTT (0.46) HTTCDK2ALDH1A1MAPTSMN1; SMN2
SCHEMBL23142017 0.80 HTT (0.46) HTTCDK2ALDH1A1MAPTSMN1; SMN2
SCHEMBL22860104 0.79 HTT (0.46) HTTCDK2ALDH1A1MAPTSMN1; SMN2
SCHEMBL23142093 0.77 HTT (0.45) HTTALDH1A1MAPTSMN1; SMN2SYK
SCHEMBL23142092 0.77 HTT (0.45) HTTALDH1A1MAPTSMN1; SMN2SYK
SCHEMBL22860671 0.77 HTT (0.46) HTTCDK2ALDH1A1MAPTSMN1; SMN2
SCHEMBL23141915 0.76 HTT (0.44) HTTALDH1A1MAPTSMN1; SMN2SYK
SCHEMBL23141916 0.76 HTT (0.44) HTTALDH1A1MAPTSMN1; SMN2SYK
SCHEMBL1521589 0.74 HTT (0.51) HTTALDH1A1MAPTSMN1; SMN2SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022187693-A1 COVALENT CDK2-BINDING COMPOUNDS FOR THERAPEUTIC PURPOSES UMBRA THERAPEUTICS INC. (US) 2022-09-09 WO disclosed