SCHEMBL24670185

SCHEMBL24670185

CC(C)(C)OC(=O)N1CC=C(c2ccc(N)cc2OC(F)(F)F)CC1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDK4 Q16654 1/20 0.51
NR1H2 P55055 1/20 0.49
HTR6 P50406 1/20 0.45
GRM1 Q13255 10/20 0.45
GRM5 P41594 9/20 0.45
JAK1 P23458 1/20 0.44
SCN9A Q15858 1/20 0.43
NAMPT P43490 1/20 0.43
CNR1 P21554 1/20 0.43
BTK Q06187 1/20 0.42
TNK2 Q07912 1/20 0.42
CCNT1 O60563 1/20 0.41
CDK9 P50750 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24670855 0.88 PDK4 (0.53) PDK4NR1H2HTR6GRM1GRM5
SCHEMBL13993115 0.86 PDK4 (0.64) PDK4HTR6GRM1GRM5JAK1
SCHEMBL29691225 0.86 PDK4 (0.64) PDK4HTR6GRM1GRM5JAK1
SCHEMBL21245850 0.85 PDK4 (0.53) PDK4NR1H2HTR6GRM1GRM5
SCHEMBL29744751 0.85 PDK4 (0.54) PDK4NR1H2HTR6GRM1GRM5
SCHEMBL6402391 0.85 PDK4 (0.54) PDK4NR1H2HTR6GRM1GRM5
SCHEMBL29744827 0.84 PDK4 (0.55) PDK4NR1H2HTR6GRM1GRM5
SCHEMBL1811363 0.84 PDK4 (0.55) PDK4NR1H2HTR6GRM1GRM5
SCHEMBL24629831 0.83 PDK4 (0.54) PDK4NR1H2HTR6GRM1GRM5
SCHEMBL31444034 0.83 PDK4 (0.54) PDK4NR1H2HTR6GRM1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed