SCHEMBL24670710

SCHEMBL24670710

O=C(Nc1ccc(Br)c(C(F)(F)F)c1)c1ccc(Br)c(F)c1

nearest known ligand 0.75

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.75
NPSR1 Q6W5P4 2/20 0.75
XBP1 P17861 1/20 0.75
MEN1 O00255 2/20 0.71
KMT2A Q03164 2/20 0.71
HTT P42858 2/20 0.71
NPC1 O15118 1/20 0.71
RAB9A P51151 1/20 0.71
LMNA P02545 2/20 0.71
SMN1; SMN2 Q16637 1/20 0.59
MAOB P27338 1/20 0.56
EPHX1 P07099 2/20 0.55
TMPRSS4 Q9NRS4 1/20 0.55
KCNQ3 O43525 2/20 0.52
KCNQ2 O43526 2/20 0.52
KCNE1 P15382 2/20 0.52
KCNQ1 P51787 2/20 0.52
ACP1 P24666 1/20 0.49
TAS2R14 Q9NYV8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803311 1.00 MAPT (0.75) MAPTNPSR1XBP1MEN1KMT2A
SCHEMBL29803393 0.96 MAPT (0.72) MAPTNPSR1XBP1MEN1KMT2A
SCHEMBL24671304 0.96 MAPT (0.72) MAPTNPSR1XBP1MEN1KMT2A
SCHEMBL24669338 0.87 MAOB (0.70) MAPTNPSR1XBP1MEN1KMT2A
SCHEMBL29803408 0.87 MAOB (0.70) MAPTNPSR1XBP1MEN1KMT2A
SCHEMBL14785061 0.86 MAPT (1.00) MAPTNPSR1XBP1MEN1KMT2A
SCHEMBL850791 0.83 MEN1 (1.00) MAPTNPSR1XBP1MEN1KMT2A
SCHEMBL24671323 0.82 MAOB (0.65) MAPTNPSR1XBP1NPC1RAB9A
SCHEMBL24670922 0.81 TP53 (0.63) MAPTMEN1KMT2ANPC1RAB9A
SCHEMBL24670881 0.80 MAOB (0.53) MAPTNPSR1XBP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed