SCHEMBL24670784

SCHEMBL24670784

COc1cc(N)c(C)cc1C1=CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK4 Q16654 1/20 0.50
GRM1 Q13255 9/20 0.48
GRM5 P41594 8/20 0.48
HTR6 P50406 1/20 0.44
JAK1 P23458 1/20 0.44
CNR1 P21554 1/20 0.42
NAMPT P43490 1/20 0.42
GABRP O00591 1/20 0.42
GABRD O14764 1/20 0.42
GABRA1 P14867 1/20 0.42
GABRB1 P18505 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42
GABRA2 P47869 1/20 0.42
GABRB2 P47870 1/20 0.42
GABRA4 P48169 1/20 0.42
GABRE P78334 1/20 0.42
GABRA6 Q16445 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18843558 0.87 PDK4 (0.50) PDK4GRM1GRM5HTR6JAK1
SCHEMBL21403965 0.87 PDK4 (0.50) PDK4GRM1GRM5HTR6JAK1
SCHEMBL1771022 0.86 PDK4 (0.51) PDK4GRM1GRM5HTR6JAK1
SCHEMBL24670953 0.86 PDK4 (0.51) PDK4GRM1GRM5HTR6JAK1
SCHEMBL24670855 0.83 PDK4 (0.53) PDK4GRM1GRM5HTR6JAK1
SCHEMBL19701842 0.83 PDK4 (0.53) PDK4GRM1GRM5HTR6JAK1
SCHEMBL1771697 0.83 PDK4 (0.48) PDK4GRM1GRM5HTR6JAK1
SCHEMBL30439968 0.82 GRM1 (0.50) PDK4GRM1GRM5HTR6JAK1
SCHEMBL21045699 0.82 GRM1 (0.50) PDK4GRM1GRM5HTR6JAK1
SCHEMBL29197044 0.82 PDK4 (0.49) PDK4GRM1GRM5HTR6JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed