SCHEMBL24671399

SCHEMBL24671399

CC(C)(C)OC(=O)N1CC=C(c2ccc(NC(=O)c3ccc(C4=CCN(C(=O)OC(C)(C)C)CC4)c(F)c3)cc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 7/20 0.60
SCN9A Q15858 1/20 0.48
PDK4 Q16654 1/20 0.47
JAK1 P23458 1/20 0.45
GRM5 P41594 4/20 0.44
GRM1 Q13255 4/20 0.44
CDK7 P50613 1/20 0.44
CDK13 Q14004 1/20 0.44
CDK12 Q9NYV4 1/20 0.44
WNT3A P56704 1/20 0.44
WDR5 P61964 2/20 0.44
PTPN2 P17706 1/20 0.43
PTPN1 P18031 1/20 0.43
PTPN6 P29350 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803696 0.94 NAMPT (0.52) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24669339 0.94 NAMPT (0.52) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL29803278 0.91 NAMPT (0.49) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24670852 0.91 NAMPT (0.49) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL29803406 0.90 NAMPT (0.49) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL29803905 0.90 NAMPT (0.49) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24669383 0.90 NAMPT (0.49) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24670039 0.90 NAMPT (0.49) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24669437 0.90 PDK4 (0.48) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24670746 0.90 NAMPT (0.61) NAMPTSCN9APDK4JAK1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed