SCHEMBL24671838

SCHEMBL24671838

CC(C)(C)OC(=O)N1CCN(CC2CCN(c3ccc([C@H]4CCC(=O)NC4=O)cc3)CC2)CC1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 11/20 0.58
CRBN Q96SW2 11/20 0.58
GPR119 Q8TDV5 7/20 0.46
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
CNR1 P21554 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24670627 1.00 DDB1 (0.58) DDB1CRBNGPR119ALDH1A1LMNA
SCHEMBL24671837 1.00 DDB1 (0.58) DDB1CRBNGPR119ALDH1A1LMNA
SCHEMBL24670555 0.96 DDB1 (0.58) DDB1CRBNGPR119ALDH1A1LMNA
SCHEMBL30801319 0.94 DDB1 (0.52) DDB1CRBNGPR119ALDH1A1LMNA
SCHEMBL24480896 0.94 DDB1 (0.54) DDB1CRBNGPR119
SCHEMBL31127609 0.91 CRBN (0.56) DDB1CRBNGPR119ALDH1A1LMNA
SCHEMBL30981278 0.90 DDB1 (0.54) DDB1CRBNGPR119CNR1
SCHEMBL21876964 0.90 DDB1 (0.67) DDB1CRBNGPR119ALDH1A1LMNA
SCHEMBL23301226 0.90 DDB1 (0.67) DDB1CRBNGPR119ALDH1A1LMNA
SCHEMBL30981193 0.88 DDB1 (0.57) DDB1CRBNGPR119ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240279202-A1 COMPOUNDS FOR INHIBITING OR DEGRADING ITK, COMPOSITIONS, COMPRISING THE SAME METHODS OF THEIR MAKING AND METHODS OF THEIR USE NURIX THERAPEUTICS, INC. 2024-08-22 US disclosed
EP-4334303-A1 COMPOUNDS FOR INHIBITING OR DEGRADING ITK, COMPOSITIONS, COMPRISING THE SAME METHODS OF THEIR MAKING AND METHODS OF THEIR USE Nurix Therapeutics, Inc. (US) 2024-03-13 EP disclosed
WO-2022235715-A1 COMPOUNDS FOR INHIBITING OR DEGRADING ITK, COMPOSITIONS, COMPRISING THE SAME METHODS OF THEIR MAKING AND METHODS OF THEIR USE NURIX THERAPEUTICS, INC. (US) 2022-11-10 WO disclosed
WO-2022235715-A1 COMPOUNDS FOR INHIBITING OR DEGRADING ITK, COMPOSITIONS, COMPRISING THE SAME METHODS OF THEIR MAKING AND METHODS OF THEIR USE NURIX THERAPEUTICS, INC. (US) 2022-11-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240279202-A1 COMPOUNDS FOR INHIBITING OR DEGRADING ITK, COMPOSITIONS, COMPRISING THE SAME METHODS OF THEIR MAKING AND METHODS OF THEIR USE ITK, NFATC1, TNIK DDB1 2514/4885CRBN 929/4885GPR119 3873/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.