SCHEMBL2467332

SCHEMBL2467332

CN(CC1CCC(C2=C3C=NC=C[N+]3(N)C(c3cccc(OCc4ccccc4)c3)=N2)CC1)C1CCNCC1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 10/20 0.38
PLAT P00750 1/20 0.37
F10 P00742 1/20 0.34
PRMT5 O14744 4/20 0.33
TNK2 Q07912 1/20 0.33
KDM1A O60341 1/20 0.33
CACNA1B Q00975 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2460188 0.87 IGF1R (0.43) IGF1RTNK2
SCHEMBL2459605 0.86 IGF1R (0.50) IGF1RTNK2
SCHEMBL2461512 0.86 IGF1R (0.40) IGF1RPRMT5TNK2
SCHEMBL2460257 0.85 IGF1R (0.40) IGF1RPLATTNK2
SCHEMBL2459995 0.85 IGF1R (0.40) IGF1RTNK2
SCHEMBL2458195 0.85 IGF1R (0.47) IGF1RPLATPRMT5TNK2
SCHEMBL2457535 0.83 IGF1R (0.38) IGF1RTNK2
SCHEMBL2460547 0.82 IGF1R (0.48) IGF1RTNK2
SCHEMBL2459690 0.82 IGF1R (0.37) IGF1RPLATTNK2
SCHEMBL2467426 0.82 TNK2 (0.40) IGF1RPRMT5TNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1675860-B1 IMIDAZO[1,5-A]PYRAZINES AS TYROSINE KINASE INHIBITORS OSI PHARM INC (US) 2011-09-21 EP claimed