SCHEMBL2467588

SCHEMBL2467588

C[C@H](CCC(=O)O)[C@H]1CC[C@H]2[C@@H]3[C@H](O)C[C@@H]4C[C@H](OC(=O)CC[C@@H](C)[C@H]5CCC6C7CCC8C[C@H](O)CC[C@]8(C)C7CC[C@@]65C)CC[C@]4(C)[C@H]3C[C@H](O)[C@]12C

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 7/20 0.72
NR1H4 Q96RI1 5/20 0.72
CYP3A4 P08684 4/20 0.72
PDE3A Q14432 2/20 0.72
LMNA P02545 3/20 0.68
MEN1 O00255 3/20 0.67
KMT2A Q03164 3/20 0.67
USP2 O75604 2/20 0.67
SLCO1B3 Q9NPD5 1/20 0.67
SLCO1B1 Q9Y6L6 1/20 0.67
SLC10A2 Q12908 2/20 0.66
TBXA2R P21731 1/20 0.66
CASP7 P55210 3/20 0.65
TDP1 Q9NUW8 3/20 0.65
TP53 P04637 2/20 0.65
MAPK1 P28482 2/20 0.65
HSD17B10 Q99714 2/20 0.65
BLM P54132 2/20 0.65
MDM4 O15151 1/20 0.65
MAPT P10636 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL246889 0.96 GPBAR1 (0.71) GPBAR1NR1H4CYP3A4PDE3ALMNA
SCHEMBL2369521 0.96 GPBAR1 (0.71) GPBAR1NR1H4CYP3A4PDE3ALMNA
SCHEMBL7546767 0.96 GPBAR1 (0.71) GPBAR1NR1H4CYP3A4PDE3ALMNA
SCHEMBL2637801 0.96 GPBAR1 (0.75) GPBAR1NR1H4CYP3A4PDE3ALMNA
SCHEMBL25791236 0.96 GPBAR1 (0.75) GPBAR1NR1H4CYP3A4PDE3ALMNA
SCHEMBL25791216 0.96 GPBAR1 (0.75) GPBAR1NR1H4CYP3A4PDE3ALMNA
SCHEMBL1287858 0.95 GPBAR1 (0.78) GPBAR1NR1H4CYP3A4PDE3ALMNA
SCHEMBL1758946 0.94 GPBAR1 (0.67) GPBAR1NR1H4CYP3A4PDE3ALMNA
SCHEMBL8646650 0.94 GPBAR1 (0.66) GPBAR1NR1H4CYP3A4PDE3ALMNA
SCHEMBL2638871 0.93 GPBAR1 (0.74) GPBAR1NR1H4CYP3A4LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367839-A2 METHODS AND COMPOSITIONS FOR INHIBITING CLOSTRIDIUM DIFFICILE SPORE GERMINATION AND OUTGROWTH Tufts University (US) 2011-09-28 EP disclosed
WO-2010062369-A2 METHODS AND COMPOSITIONS FOR INHIBITING CLOSTRIDIUM DIFFICILE SPORE GERMINATION AND OUTGROWTH TUFTS UNIVERSITY (US) 2010-06-03 WO disclosed