SCHEMBL24676930

SCHEMBL24676930

CN(C)Cc1nc(C(F)(F)F)c(-c2ccnc(NC3CCN(S(C)(=O)=O)CC3)n2)s1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 5/20 0.52
CDK2 P24941 13/20 0.46
CCNE1 P24864 8/20 0.46
PTK2 Q05397 1/20 0.44
CCND1 P24385 10/20 0.42
CDK6 Q00534 10/20 0.42
CDK4 P11802 8/20 0.41
CCND3 P30281 7/20 0.41
CDK1 P06493 6/20 0.41
CCNB1 P14635 6/20 0.41
CCNA2 P20248 5/20 0.41
CDK7 P50613 4/20 0.41
CCNH P51946 4/20 0.41
CCNT1 O60563 3/20 0.41
CDK9 P50750 3/20 0.41
IDH1 O75874 1/20 0.41
IDH2 P48735 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29754851 1.00 IKBKB (0.52) IKBKBCDK2CCNE1PTK2CCND1
SCHEMBL29754874 0.90 IKBKB (0.54) IKBKBCDK2CCNE1PTK2CCND1
SCHEMBL24675988 0.90 IKBKB (0.54) IKBKBCDK2CCNE1PTK2CCND1
SCHEMBL24677023 0.87 IKBKB (0.52) IKBKBCDK2CCNE1PTK2CCND1
SCHEMBL24676939 0.86 CDK4 (0.42) IKBKBCDK2CCND1CDK6CDK4
SCHEMBL24676458 0.85 IKBKB (0.49) IKBKBCDK2CCNE1PTK2CCND1
SCHEMBL24675961 0.84 IKBKB (0.58) IKBKBCDK2CCNE1CCND1CDK6
SCHEMBL29755006 0.84 IKBKB (0.56) IKBKBCDK2CCNE1CCND1CDK6
SCHEMBL24676704 0.84 IKBKB (0.56) IKBKBCDK2CCNE1CCND1CDK6
SCHEMBL24676765 0.84 CDK2 (0.54) CDK2CCNE1PTK2CCND1CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022155941-A1 CDK2 INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2022-07-28 WO disclosed