SCHEMBL24680708

SCHEMBL24680708

CC(C)(C)OC(=O)N1CCN(c2ccc(-c3cnc(N)c(-c4ccc5c(c4)CCNC5=O)c3)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.47
FYN P06241 7/20 0.46
TGFBR1 P36897 8/20 0.45
ACVR1 Q04771 7/20 0.45
ATR Q13535 1/20 0.43
ALK Q9UM73 1/20 0.42
PIK3CA P42336 1/20 0.42
RIPK2 O43353 1/20 0.42
NOD2 Q9HC29 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29914385 1.00 MAPK1 (0.47) MAPK1FYNTGFBR1ACVR1ATR
SCHEMBL29914600 0.88 MAPK1 (0.52) MAPK1FYNTGFBR1ACVR1RIPK2
SCHEMBL24680722 0.88 MAPK1 (0.52) MAPK1FYNTGFBR1ACVR1RIPK2
SCHEMBL24681143 0.88 MAPK1 (0.42) MAPK1PIK3CA
SCHEMBL29914518 0.88 MAPK1 (0.42) MAPK1PIK3CA
SCHEMBL29964242 0.87 MAPK1 (0.54) MAPK1
SCHEMBL24680920 0.86 MAPK1 (0.47) MAPK1FYNTGFBR1ACVR1RIPK2
SCHEMBL29914464 0.86 MAPK1 (0.47) MAPK1FYNTGFBR1ACVR1RIPK2
SCHEMBL31079257 0.85 SMARCA2 (0.40) MAPK1TGFBR1ACVR1ATRALK
SCHEMBL29964997 0.85 RET (0.40) MAPK1TGFBR1ACVR1ATRALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022226667-A1 SUBSTITUTED AMINO PYRIDINE COMPOUNDS AS INHIBITORS OF THE HAEMATOPOIETIC PROGENITOR KINASE 1 (HPK1) ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR) (CA) 2022-11-03 WO disclosed