SCHEMBL24697153

SCHEMBL24697153

CCCC(CC)C(OCC)c1ccccn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 5/20 0.43
KCNH2 Q12809 4/20 0.43
CYP2D6 P10635 4/20 0.41
KCNE1 P15382 1/20 0.41
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TSHR P16473 2/20 0.38
CHRM2 P08172 5/20 0.37
SLC6A2 P23975 5/20 0.37
SLC6A4 P31645 5/20 0.37
SCN1A P35498 2/20 0.37
SCN2A Q99250 2/20 0.37
SCN3A Q9NY46 2/20 0.37
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CHRM1 P11229 3/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21742015 0.79 KCNA5 (0.45) KCNA5KCNH2CYP2D6KCNE1MEN1
SCHEMBL20278799 0.78 KCNA5 (0.41) KCNA5KCNH2CYP2D6KCNE1MEN1
SCHEMBL21742251 0.76 KCNA5 (0.45) KCNA5KCNH2CYP2D6KCNE1MEN1
SCHEMBL22131652 0.75 KCNA5 (0.40) KCNA5KCNH2CYP2D6KCNE1MEN1
SCHEMBL3804481 0.74 KCNA5 (0.44) KCNA5KCNH2CYP2D6KCNE1MEN1
SCHEMBL21742078 0.74 KCNA5 (0.50) KCNA5KCNH2CYP2D6KCNE1MEN1
SCHEMBL15704684 0.73 KCNA5 (0.49) KCNA5KCNH2CYP2D6KCNE1MEN1
SCHEMBL28012567 0.73 KCNA5 (0.49) KCNA5KCNH2CYP2D6KCNE1MEN1
SCHEMBL21742062 0.72 KCNA5 (0.49) KCNA5KCNH2CYP2D6KCNE1MEN1
SCHEMBL21742012 0.72 KCNA5 (0.49) KCNA5KCNH2CYP2D6KCNE1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3412663-B1 NITROGEN-CONTAINING HETEROCYCLE AND CARBOCYCLE DERIVATIVES HAVING TRKA INHIBITORY ACTIVITY SHIONOGI & CO (JP) 2022-09-07 EP disclosed