SCHEMBL2471192

SCHEMBL2471192

CS(=O)(=O)N(CCO)c1cn2ncc(C(=O)O)c2c(-c2ccc(F)cc2)c1-c1cccc(C(=O)NC2(c3ccccn3)CC2)c1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.37
NR1I2 O75469 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C8 P10632 1/20 0.37
ACKR3 P25106 1/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
DGAT2 Q96PD7 1/20 0.31
ADRB1 P08588 1/20 0.31
CCR1 P32246 1/20 0.31
LIPG Q9Y5X9 1/20 0.31
RET P07949 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2466024 0.81 CYP3A4 (0.40) KCNH2NR1I2CYP3A4CYP2C8ACKR3
SCHEMBL1935953 0.78 CYP2C8 (0.46) KCNH2NR1I2CYP3A4CYP2C8
SCHEMBL1936441 0.77 CYP3A4 (0.40) KCNH2NR1I2CYP3A4CYP2C8ACKR3
SCHEMBL2142749 0.74 CYP3A4 (0.62) KCNH2NR1I2CYP3A4CYP2C8
SCHEMBL2464251 0.71 CYP2C8 (0.47) KCNH2NR1I2CYP3A4CYP2C8
SCHEMBL1936876 0.68 PTPN1 (0.35) CYP3A4
SCHEMBL2991655 0.66 CYP3A4 (0.39) KCNH2NR1I2CYP3A4CYP2C8ACKR3
SCHEMBL1936957 0.65 EPHB3 (0.41) KCNH2NR1I2CYP3A4CYP2C8DGAT2
SCHEMBL1937048 0.65 CYP2C8 (0.53) KCNH2NR1I2CYP3A4CYP2C8ACKR3
SCHEMBL2143033 0.65 CYP3A4 (0.60) CYP3A4CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2545050-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C Bristol-Myers Squibb Company (US) 2013-01-16 EP disclosed
WO-2011112186-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2011-09-15 WO disclosed